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A prerequisite for rapid renal elimination is a hepatic conjugation reaction (p. 38), mainly with glycine (> salicyluric acid) and glucuronic acid. At high dosage, the conjugation may become rate limiting. Elimination now increasingly depends on unchanged salicylate, which is excreted only slowly. Group-specific adverse effects can be attributed to inhibition of cyclooxygenase (B).
In addition, patients exhibit delusional paranoia (persecution mania) or hallucinations (fearfulness hearing of voices). Contrasting these “positive” symptoms, the so-called “negative” symptoms, viz. , poverty of thought, social withdrawal, and anhedonia, assume added importance in determining the severity of the disease. |
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